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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Ponatinib Influence on protein activity Western Blot 10.00 µM IMR-32 Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity Western Blot 10.00 µM NGP Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity Western Blot 10.00 µM NB-19 Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity Western Blot 10.00 µM SH-SY5Y Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity Western Blot 10.00 µM SK-N-AS Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity Western Blot 10.00 µM LA-N6 Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 2.00 µM NGP Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 5.00 µM NGP Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 10.00 µM NGP Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 20.00 µM NGP Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 2.00 µM SH-SY5Y Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 5.00 µM SH-SY5Y Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 10.00 µM SH-SY5Y Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in presence of bFGF Western Blot 20.00 µM SH-SY5Y Homo sapiens p-STAT3 (Y705)
Ponatinib Influence on protein activity in tumor tissue Western Blot 15.00 mg/kg NB-19 (xenograft) Mus musculus NCr nude mice p-STAT3 (Y705)